Thiazolidinone motif in anticancer drug discovery. Experience of DH LNMU medicinal chemistry scientific group RB Lesyk, BS Zimenkovsky, DV Kaminskyy, AP Kryshchyshyn, ... Âiopolymers and Cell, 2011 | 126 | 2011 |
Synthesis of 5-arylidene-2-amino-4-azolones and evaluation of their anticancer activity I Subtel’na, D Atamanyuk, E Szymańska, K Kieć-Kononowicz, ... Bioorganic & medicinal chemistry 18 (14), 5090-5102, 2010 | 123 | 2010 |
Synthesis and antiinflammatory activity of some 2-arylamino-2-thiazoline-4-ones Roman Lesyk, Boris Zimenkovsky, Ivanna Subtelna, Igor Nektegayev, Gennadij ... Acta poloniae pharmaceutica 60 (6), 457-466, 2003 | 42 | 2003 |
Synthesis and evaluation of anticancer activity of 5-ylidene-4-aminothiazol-2 (5H)-one derivatives D Kaminskyy, I Subtel’na, B Zimenkovsky, O Karpenko, A Gzella, R Lesyk Medicinal Chemistry 11 (6), 517-530, 2015 | 34 | 2015 |
Anticancer potential of 4-azolidones and related heterocycles R Lesyk, B Zimenkovsky, D Kaminskyy, S Holota, D Atamanyuk, ... Ann. Univ. Mariae Curie-Sklodowska. Med 19 (1), 107-110, 2006 | 18 | 2006 |
The structure – anti-inflammatory activity relationship among thiazolidones: conclusion from scientific programme IC B. Zimenkovsky, O.Vladzimirska, R.Lesyk, I. Nektegayev, S. Golota Journal of Pharmacy and Pharmacology 51 (3), 264, 1999 | 18 | 1999 |
One-Pot Synthesis of 5-Ene-4-aminothiazol-2 (5H)-ones and Chromeno [2, 3-d] thiazol-2-ones D Kaminskyy, I Subtel’na, A Pyrih, D Shtoyko, A Susel, A Gzella, R Lesyk Synlett 28 (07), 811-814, 2017 | 11 | 2017 |
5‐Arylidene‐2‐(4‐hydroxyphenyl)aminothiazol‐4(5H)‐ones with selective inhibitory activity against some leukemia cell lines I Subtelna, A Kryshchyshyn‐Dylevych, R Jia, M Lelyukh, A Ringler, ... Archiv der Pharmazie 354 (4), 2000342, 2021 | 8 | 2021 |
Anticancer 5‐arylidene‐2‐(4‐hydroxyphenyl)aminothiazol‐4(5H)‐ones as tubulin inhibitors J Rehulka, I Subtelna, A Kryshchyshyn‐Dylevych, A Cherniienko, ... Archiv der Pharmazie 355 (12), 2200419, 2022 | 7 | 2022 |
Ñó÷àñí³ ï³äõîäè äî ìîäåëþâàííÿ ë³êàðñüêèõ çàñîá³â ÐÁ Ëåñèê, ÁÏ Ãðîìîâèê, Ä Àòàìàíþê, ²Þ Ñóáòåëüíà, ²² Ñîðîíîâè÷ Ôàðìàö. æóðí, 33-39, 2002 | 5 | 2002 |
Anticancer cytotoxicity of indole-thiazolidinone hybrids, in silico study of mechanisms of their action AP Kryshchyshyn-Dylevych, IY Subtelna, NS Finiuk, L Radko, ... Biopolymers and Cell 38 (4), 257-277, 2022 | 1 | 2022 |
In sIlIco identification and biochemical validation of plausible molecular targets of 4-thiazolidinone derivative les-3833 as a potential anticancer agent RL L. KîbylinsKa, D. Khylyuk, I. Subtelna, M. Kitsera Ukrainian Biochemical Journal 93 (2), 7-22, 2021 | 1 | 2021 |
Synthesis and antitumor activity evaluation of new 2-(4-alkoxyphenylamino) thiazol-4 (5H)-onesderivatives I Subtel'na, B Zimenkovsky, R Lesyk Pharmacia 23 (3), 231-235, 2010 | 1 | 2010 |
Ïðîòèïóõëèííà öèòîòîêñè÷í³ñòü ³íäîë-ò³àçîë³äèíîíîâèõ ã³áðèä³â òà in silico äîñë³äæåííÿ ìåõàí³çìó ¿õíüî¿ ä³¿ ÀÏ Êðèùèøèí-Äèëåâè÷, ²Þ Ñóáòåëüíà, ÍÑ Ô³íþê, Ë Ðàäêî, ... Biopolymers and Cell 38 (4), 257-277, 2022 | | 2022 |
Ñèíòåç, ïðåâðàùåíèÿ è áèîëîãè÷åñêàÿ àêòèâíîñòü ôóíêöèîíàëüíîçàìåùåííûõ 2-àìèíî-2-òèàçîëèí-4-îíîâ è 2(4)-èìèíî-4(2)-òèàçîëèäèíîíîâ Ä.ß. Ãàâðèëþê, È.Þ. Ñóáòåëüíàÿ, Á.Ñ. Çèìåíêîâñêèé “Õèìèÿ è áèîëîãè÷åñêàÿ àêòèâíîñòü àçîëîâ” (Èçáðàííûå îáçîðû) ïîä ðåäàêöèåé  …, 2014 | | 2014 |
Rational design of potential anticancer" drug-like" molecules based on 4-azoldinone scaffold R Lesyk, B Zimenkovsky, D Kaminskyy, D Havryluk, D Atamanyuk, ... EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS 40, 109-109, 2011 | | 2011 |
Ò³àçîë³äèíîíè ÿê ëåéòìîòèâ ó ñòâîðåíí³ ïðîòèðàêîâèõ ë³êàðñüêèõ çàñîá³â. Äîñâ³ä íàóêîâî¿ ãðóïè ç ìåäè÷íî¿ õ³ì³¿ ËÍÌÓ ³ìåí³ Äàíèëà Ãàëèöüêîãî ÐÁ Ëåñèê, ÁÑ Ç³ìåíêîâñüêèé, Ä Êàì³íñüêèé, ÀÏ Êðèùèøèí, ... Biopolymers and Cell 27 (2), 107-117, 2011 | | 2011 |
RECOOP Biopolymers and Cell SG Vari | | 2011 |
ÑÈÍÒÅÇ È ÈÇÓ×ÅÍÈÅ ÏÐÎÒÈÂÎÎÏÓÕÎËÅÂÎÉ ÀÊÒÈÂÍÎÑÒÈ ÏÐÎÈÇÂÎÄÍÛÕ 2-(4-ÀËÊÎÊÑÈ-ÔÅÍÈËÀÌÈÍÎ) ÒÈÀÇÎË-4 (5Í)-ÎÍΠ²Þ Ñóáòåëüíà, ÁÑ Ç³ìåíêîâñüêèé, ÐÁ Ëåñèê Æóðíàë îðãàí³÷íî¿ òà ôàðìàöåâòè÷íî¿ õ³ì³¿ 8 (3), 58-64, 2010 | | 2010 |
ÑÈÍÒÅÇ 5-ÀÐÈ˲ÄÅÍÏÎÕ²ÄÍÈÕ (2-ÌÅÒÈË-4-ÎÊÑÈ-5-²ÇÎÏÐÎϲËÔÅͲËÀ̲ÍÎ) Ò²ÀÇÎËÎͲ ÒÀ ÂÈÂ×ÅÍÍß ¯Õ ÏÐÎÒÈÏÓÕËÈÍÍί ÀÊÒÈÂÍÎÑÒ² ²Þ Ñóáòåëüíà, ÁÑ Ç³ìåíêîâñüêèé, À Ãçåëëÿ, ÃÌ Ñåìåíö³â, ... Êë³í³÷íà ôàðìàö³ÿ, ôàðìàêîòåðàï³ÿ òà ìåäè÷íà ñòàíäàðòèçàö³ÿ, 93, 2010 | | 2010 |