Heterocyclization of N-(1-chloro-2, 2, 2-trifluoroethylidene) carbamates with β-enaminoesters—a novel synthetic strategy to functionalized trifluoromethylated pyrimidines VA Sukach, VM Tkachuk, EB Rusanov, GV Röschenthaler, MV Vovk Tetrahedron 68 (40), 8408-8415, 2012 | 39 | 2012 |
Development of an efficient route to CF 3-substituted pyrrolopyrimidines through understanding the competition between Michael and aza-Henry reactions VM Tkachuk, VA Sukach, KV Kovalchuk, MV Vovk, VG Nenajdenko Organic & Biomolecular Chemistry 13 (5), 1420-1428, 2015 | 20 | 2015 |
Aza‐Henry Reaction with CF3‐Ketimines: An Efficient Approach to Trifluoromethylated β‐Nitroamines, 1,2‐Diamines, α‐Aminooximes, and Imidazolidinones IV Kutovaya, OI Shmatova, VM Tkachuk, NV Melnichenko, MV Vovk, ... European Journal of Organic Chemistry 2015 (30), 6749-6761, 2015 | 18 | 2015 |
Control of Regio‐ and Enantioselectivity in the Asymmetric Organocatalytic Addition of Acetone to 4‐(Trifluoromethyl)pyrimidin‐2(1H)‐ones VA Sukach, VM Tkachuk, VM Shoba, VV Pirozhenko, EB Rusanov, ... European Journal of Organic Chemistry 2014 (7), 1452-1460, 2014 | 17 | 2014 |
Asymmetric organocatalytic mannich reaction of 1-aryl-2, 2, 2-trifluoroethylidenecarbamic acid derivatives with acetone NM Golovach, VN Tkachuk, VA Sukach, MV Vovk Russian Journal of Organic Chemistry 48, 1187-1190, 2012 | 14 | 2012 |
Synthesis of Trifluoromethylated Analogues of 4, 5‐Dihydroorotic Acid VA Sukach, AA Resetnic, VM Tkachuk, Z Lin, U Kortz, MV Vovk, ... European Journal of Organic Chemistry 2015 (6), 1290-1301, 2015 | 10 | 2015 |
Convenient synthesis of 4-pyridinyloxy-modified imidazo [2, 1-b][1, 3] thiazines as potential anti-inflammatory agents N Slyvka, L Saliyeva, S Holota, V Tkachuk, A Vaskevych, R Vaskevych, ... Biointerface Res. Appl. Chem 13 (1), 6033-6044, 2023 | 7 | 2023 |
The addition of β-ketoacids to 4-(trifluoromethyl)pyrimidin- 2(1Н)-ones with decarboxylation: an effective method for the synthesis of 4-(2-oxoalkyl)-6-(trifluoromethyl … VM Tkachuk, SV Mel’nikov, VA Sukach, MV Vovk Chemistry of Heterocyclic Compounds 53, 1124-1127, 2017 | 7 | 2017 |
Chan–Evans–Lam N1-(het) arylation and N1-alkеnylation of 4-fluoroalkylpyrimidin-2 (1H)-ones VM Tkachuk Beilstein Journal of Organic Chemistry 16 (1), 2304-2313, 2020 | 6 | 2020 |
Study of regioselectivity in cyanomethylation of 4-(trifluoromethyl)pyrimidin-2(1Н)-ones VM Tkachuk, SV Melnykov, AV Vorobei, VA Sukach, MV Vovk Chemistry of Heterocyclic Compounds 55, 66-71, 2019 | 5 | 2019 |
Oxidative Nef reaction of trifluoromethylated 2-nitroalkanamines IV Kutovaya, OI Shmatova, VM Tkachuk, VA Sukach, MV Vovk, ... Mendeleev Communications 26 (6), 511-512, 2016 | 4 | 2016 |
N-Benzyloxycarbonyl-2, 2, 2-trifluoroacetimidoyl chloride-A convenient reagent for the synthesis of 2-trifluoromethyl-4 H-pyrido [1, 2-a][1, 3, 5] triazin-4-one. N Mel'nichenko, V Tkachuk, E Rusanov, V Sukach, V Boiko, M Vovk Russian Journal of Organic Chemistry 49 (1), 2013 | 4 | 2013 |
Modern Approaches to Synthetic Design of Chiral α-Tertiary Amines Based on Trifluoromethylcontaining Ketimines: A Review VA Sukach, VM Tkachuk, I Gillaizeau, MV Vovk Theoretical and Experimental Chemistry 57 (6), 387-420, 2022 | 2 | 2022 |
Sulfones of Pyridinyloxy-Substituted Imidazo [2, 1-b][1, 3] thiazines: Synthesis, Anti-Inflammatory Activity Evaluation In Vivo and Docking Studies N Slyvka, L Saliyeva, S Holota, D Khyluk, V Tkachuk, M Vovk Letters in Drug Design & Discovery 20 (11), 1867-1875, 2023 | 1 | 2023 |
Hydroaminoalkyl Functionalization of Pyrimidin‐2(1H)‐ones by Visible Light Organophotocatalysis: A Radical Approach to Biginelli‐Type Dihydropyrimidines O Lukianov, V Tkachuk, S Shishkina, L Lachmann, O Vadzyuk, P Borysko, ... Advanced Synthesis & Catalysis 365 (20), 3484-3492, 2023 | 1 | 2023 |
Синтез та деякі перетворення алкіл N-(2-арил-3-нітро-1, 1, 1-трифторопропан-2-іл) карбаматів VM Tkachuk, NV Melnichenko, KV Kovalchuk, VA Sukach, MV Vovk, ... Journal of Organic and Pharmaceutical Chemistry 12 (4 (48)), 71-76, 2014 | 1 | 2014 |
Synthesis, Chemical and Biological Properties of Trifluoromethylated Pyrimidin-2-ones (thiones) and Their Fused Analogues VM Shoba, VM Tkachuk, VA Sukach, MV Vovk Targets in Heterocyclic Systems, 147, 2013 | 1 | 2013 |
An Efficient Synthesis of PARP Inhibitors Containing a 4-Trifluoromethyl Substituted 3, 6, 7, 7a-Tetrahydro-1H-pyrrolo [3, 4-d] pyrimidine-2, 5-dione Scaffold O Lukianov, VM Tkachuk, DS Stepanova, I Gillaizeau, VA Sukach Journal of Organic and Pharmaceutical Chemistry 21 (4), 18-26, 2023 | | 2023 |
Синтез 3-арил-3-трифторометил-2, 3-дигідро-1Н-піролізин-1-онів СВ Мельников, ВМ Ткачук, АМ Грозав, І Жілазо, ВА Сукач Журнал органічної та фармацевтичної хімії, 13-19, 2019 | | 2019 |
Трифторометиловмісні 3, 4-дигідропіримідин-2-они та їх конденсовані аналоги SV Mel’nikov, VM Tkachuk, VA Sukach, MV Vovk Journal of Organic and Pharmaceutical Chemistry 16 (3 (63)), 3-23, 2018 | | 2018 |