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Volodymyr Bdzhola
Volodymyr Bdzhola
Подтвержден адрес электронной почты в домене imbg.org.ua - Главная страница
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Процитировано
Год
Evaluation of 3-Carboxy-4(1H)-quinolones as Inhibitors of Human Protein Kinase CK2
AG Golub, OY Yakovenko, VG Bdzhola, VM Sapelkin, P Zien, ...
Journal of medicinal chemistry 49 (22), 6443-6450, 2006
872006
Synthesis and biological evaluation of substituted (thieno [2, 3-d] pyrimidin-4-ylthio) carboxylic acids as inhibitors of human protein kinase CK2
AG Golub, VG Bdzhola, NV Briukhovetska, AO Balanda, OP Kukharenko, ...
European journal of medicinal chemistry 46 (3), 870-876, 2011
792011
Identification of 3H-Naphtho[1,2,3-de]quinoline-2,7-diones as Inhibitors of Apoptosis Signal-Regulating Kinase 1 (ASK1)
GP Volynets, MO Chekanov, AR Synyugin, AG Golub, OP Kukharenko, ...
Journal of medicinal chemistry 54 (8), 2680-2686, 2011
632011
Evaluation of 4, 5, 6, 7-tetrahalogeno-1H-isoindole-1, 3 (2H)-diones as inhibitors of human protein kinase CK2
AG Golub, OY Yakovenko, AO Prykhod'Ko, SS Lukashov, VG Bdzhola, ...
Biochimica et Biophysica Acta (BBA)-Proteins and Proteomics 1784 (1), 143-149, 2008
612008
Design, synthesis and biological evaluation of N-phenylthieno [2, 3-d] pyrimidin-4-amines as inhibitors of FGFR1
AA Gryshchenko, VG Bdzhola, AO Balanda, NV Briukhovetska, IM Kotey, ...
Bioorganic & Medicinal Chemistry 23 (9), 2287-2293, 2015
392015
Discovery and characterization of synthetic 4′-hydroxyflavones—New CK2 inhibitors from flavone family
AG Golub, VG Bdzhola, OV Ostrynska, IV Kyshenia, VM Sapelkin, ...
Bioorganic & medicinal chemistry 21 (21), 6681-6689, 2013
392013
Structure-based discovery of novel flavonol inhibitors of human protein kinase CK2
AG Golub, VG Bdzhola, YV Kyshenia, VM Sapelkin, AO Prykhod’ko, ...
Molecular and cellular biochemistry 356 (1), 107-115, 2011
362011
Discovery of potent anti-tuberculosis agents targeting leucyl-tRNA synthetase
OI Gudzera, AG Golub, VG Bdzhola, GP Volynets, SS Lukashov, ...
Bioorganic & Medicinal Chemistry 24 (5), 1023-1031, 2016
342016
Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1, 5-dihydro-pyrrol-2-one
SA Starosyla, GP Volynets, SS Lukashov, OB Gorbatiuk, AG Golub, ...
Bioorganic & Medicinal Chemistry 23 (10), 2489-2497, 2015
322015
Kirchhoff atomic charges fitted to multipole moments: implementation for a virtual screening system
O Yakovenko, AA Oliferenko, VG Bdzhola, VA Palyulin, NS Zefirov
Journal of computational chemistry 29 (8), 1332-1343, 2008
322008
Design, synthesis and evaluation of 3-quinoline carboxylic acids as new inhibitors of protein kinase CK2
AR Syniugin, OV Ostrynska, MO Chekanov, GP Volynets, SA Starosyla, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup4), 160-169, 2016
282016
Treatment of cultured human astrocytes and vascular endothelial cells with protein kinase CK2 inhibitors induces early changes in cell shape and cytoskeleton
AA Kramerov, AG Golub, VG Bdzhola, SM Yarmoluk, K Ahmed, M Bretner, ...
Molecular and cellular biochemistry 349 (1), 125-137, 2011
282011
Design and synthesis of novel protein kinase CK2 inhibitors on the base of 4-aminothieno [2, 3-d] pyrimidines
OV Ostrynska, AO Balanda, VG Bdzhola, AG Golub, IM Kotey, ...
European Journal of Medicinal Chemistry 115, 148-160, 2016
252016
A note of caution on the role of halogen bonds for protein kinase/inhibitor recognition suggested by high-and low-salt CK2α complex structures
B Guerra, N Bischoff, VG Bdzhola, SM Yarmoluk, OG Issinger, AG Golub, ...
ACS Chemical Biology 10 (7), 1654-1660, 2015
252015
Rational design of apoptosis signal-regulating kinase 1 inhibitors: discovering novel structural scaffold
GP Volynets, VG Bdzhola, AG Golub, AR Synyugin, MA Chekanov, ...
European Journal of Medicinal Chemistry 61, 104-115, 2013
242013
Identification of novel PARP-1 inhibitors by structure-based virtual screening
K Hannigan, SS Kulkarni, VG Bdzhola, AG Golub, SM Yarmoluk, ...
Bioorganic & medicinal chemistry letters 23 (21), 5790-5794, 2013
232013
Design, synthesis and biological evaluation of 5-amino-4-(1H-benzoimidazol-2-yl)-phenyl-1, 2-dihydro-pyrrol-3-ones as inhibitors of protein kinase FGFR1
AA Gryshchenko, SS Tarnavskiy, KV Levchenko, VG Bdzhola, ...
Bioorganic & Medicinal Chemistry 24 (9), 2053-2059, 2016
192016
The new method of distribution integrals evaluations for high throughput virtual screening
OY Yakovenko, AA Oliferenko, AG Golub, VG Bdzhola, SM Yarmoluk
Ukr. Bioorg. Acta 1, 52-62, 2007
192007
Identification of Mycobacterium tuberculosis leucyl-tRNA synthetase (LeuRS) inhibitors among the derivatives of 5-phenylamino-2H-[1,2,4]triazin-3-one
OI Gudzera, AG Golub, VG Bdzhola, GP Volynets, OP Kovalenko, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup2), 201-207, 2016
172016
Electrochemical screening of the indole/quinolone derivatives as potential protein kinase CK2 inhibitors
S Martić, S Tackenburg, Y Bilokin, A Golub, V Bdzhola, S Yarmoluk, ...
Analytical biochemistry 421 (2), 617-621, 2012
172012
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