Підписатись
Antypenko Oleksii Mykolayovych/Антипенко Олексій Миколайович/Антипенко Алексей Николаевич
Antypenko Oleksii Mykolayovych/Антипенко Олексій Миколайович/Антипенко Алексей Николаевич
Zaporizhzhia State Medical University/Запорізький Державний медичний університет
Підтверджена електронна адреса в zsmu.zp.ua - Домашня сторінка
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Synthesis and biological activity of novel N-cycloalkyl-(cycloalkylaryl)-2-[(3-R-2-oxo-2H-[1, 2, 4] triazino [2, 3-c] quinazoline-6-yl) thio] acetamides
GG Berest, OY Voskoboynik, SI Kovalenko, OM Antypenko, IS Nosulenko, ...
European journal of medicinal chemistry 46 (12), 6066-6074, 2011
722011
Synthesis and anticancer activity of 2-(alkyl-, alkaryl-, aryl-, hetaryl-)-[1, 2, 4] triazolo [1, 5-c] quinazolines
SI Kovalenko, LM Antypenko, AK Bilyi, SV Kholodnyak, OV Karpenko, ...
Scientia pharmaceutica 81 (2), 359-392, 2013
462013
Design and evaluation of novel antimicrobial and anticancer agents among tetrazolo [1, 5-c] quinazoline-5-thione S-derivatives
LM Antypenko, SI Kovalenko, OM Antypenko, AM Katsev, OM Achkasova
Scientia pharmaceutica 81 (1), 15-42, 2013
332013
Novel N-aryl(alkaryl)-2-[(3-R-2-oxo-2H-[1,2,4]triazino[2,3-c]quinazoline-6-yl)thio]acetamides: synthesis, cytotoxicity, anticancer activity, COMPARE analysis and …
SI Kovalenko, IS Nosulenko, AY Voskoboynik, GG Berest, LN Antipenko, ...
Medicinal Chemistry Research 22, 2610-2632, 2013
302013
Substituted 2-[(2-oxo-2H-[1, 2, 4] triazino [2, 3-c] quinazolin-6-yl) thio] acetamides with thiazole and thiadiazole fragments: synthesis, physicochemical properties …
SI Kovalenko, IS Nosulenko, AY Voskoboynik, GG Berest, LN Antypenko, ...
Scientia Pharmaceutica 80 (4), 837-866, 2012
302012
Design, Synthesis and Anti-inflammatory Activity of Derivatives 10-R-3-Aryl-6, 7-dihydro-2H-[1, 2, 4] triazino [2, 3-c] quinazolin-2-ones of Spiro-fused Cyclic Frameworks
O Kolomoets, O Voskoboynik, O Antypenko, G Berest, I Nosulenko, ...
Slovensko kemijsko društvo, 2017
282017
Synthesis of new 6-{[ω-(dialkylamino (heterocyclyl) alkyl] thio}-3-R-2H-[1, 2, 4] triazino [2, 3-c] quinazoline-2-ones and evaluation of their anticancer and antimicrobial …
GG Berest, OY Voskoboynik, SI Kovalenko, IS Nosulenko, LM Antypenko, ...
Scientia Pharmaceutica 80 (1), 37-66, 2012
262012
Synthesis, spectroscopic characterization, X-ray structure, and in vivo neurotropic activity of new 1, 5-benzodiazepin-2-ones
AA Gaponov, ET Zlenko, SV Shishkina, OV Shishkin, OM Antypenko, ...
Medicinal Chemistry Research 25, 1768-1780, 2016
232016
Directed search of anti-inflammatory agents among (3H-quinazoline-4-ylidene) hydrazides of N-protected amino acids and their heterocyclization products
Y Martynenko, O Antypenko, I Nosulenko, G Berest, S Kovalenko
Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry (Formerly …, 2020
202020
Potential of N-aryl (benzyl, heteryl)-2-(tetrazolo [1, 5-c] quinazolin-5-ylthio) acetamides as anticancer and antimicrobial agents
OM Antypenko, LM Antypenko, SI Kovalenko, AM Katsev, OM Achkasova
Arabian Journal of Chemistry 9 (6), 792-805, 2016
202016
Synthesis, Anticancer, and QSAR Studies of 2‐Alkyl(aryl,hetaryl)quinazolin‐4(3H)‐thione's and [1,2,4]Triazolo[1,5‐c]quinazoline‐2‐thione's Thioderivatives
OM Antypenko, SI Kovalenko, OV Karpenko, VO Nikitin, LM Antypenko
Helvetica Chimica Acta 99 (8), 621-631, 2016
172016
Synthesis and hydrolytic cleavage of tetrazolo [1, 5-c] quinazolines
OM Antypenko, SI Kovalenko, OV Karpenko
Synthetic Communications 46 (6), 551-555, 2016
172016
Substituted 3-R-2, 8-Dioxo-7, 8-dihydro-2H-pyrrolo [1, 2-a][1, 2, 4] triazino [2, 3-c] quinazoline-5a (6H) carboxylic Acids and their Salts–a Promising Class of Anti …
V Stavytskyi, O Antypenko, I Nosulenko, G Berest, O Voskoboinik, ...
Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry (Formerly …, 2021
92021
Search for compounds with hypoglycemic activity in the series of 1-(2-(1H-Tetrazol-5-yl)-R1-Phenyl)-3-R2-phenyl (ethyl) ureas and R1-Tetrazolo [1, 5-c] quinazolin-5 (6H)-ones
OM Antypenko, SI Kovalenko, GО ZHERNOVA
Scientia Pharmaceutica 84 (2), 233-254, 2016
92016
5, 6-Dihydro-(1, 2, 4) triazolo (1, 5-с) quinazolines. Message 2.(5+ 1)-Cyclocondensation of (2-(3-aryl-1H-1, 2, 4-triazol-5-yl) phenyl) amines with aliphatic and aromatic ketones
SV Kholodnyak, KP Schabelnyk, OY Voskoboynik, OM Antypenko, ...
Харків: НФаУ, 2016
72016
Investigation of actoprotective activity in a range of 6-NR-tetrazolo/1, 5-c/quinazolin-5 (6H)-ones
OM Antypenko, SI Kovalenko, SD Trzhetsinsky
Запорожский медицинский журнал, 81-84, 2016
72016
Tandem heterocyclization of 2‐(azolyl‐(azinyl‐)) anilines as an efficient method for preparation of substituted pyrrolo [1, 2‐a] azolo‐(azino‐)[c] quinazolines
V Stavytskyi, O Voskoboinik, O Antypenko, N Krasovska, K Shabelnyk, ...
Journal of Heterocyclic Chemistry 57 (3), 1249-1260, 2019
62019
Synthesis of new 6-{thio}-3-R-2H-triazino quinazoline-2-ones and evaluation of their anticancer and antimicrobial activities
GG Berest, OY Voskoboynik, SI Kovalenko, IS Nosulenko, LM Antypenko, ...
Sci. Pharm 80 (1), 37, 2012
62012
Synthesis and Hypolipidemic Activity of New 6,6‐Disubstituted 3‐R‐6,7‐Dihydro‐2H‐[1,2,4]triazino[2,3‐c]quinazolin‐2‐Ones
ОY Voskoboynik, OS Kolomoets, OM Antypenko, GО Zhernova, ...
Journal of Heterocyclic Chemistry 55 (1), 318-325, 2018
52018
Synthesis of 6-NR-Tetrazolo [1, 5-c] quinazolin-5 (6H)-ones and Their Anticancer Activity
O Antypenko, S Kovalenko
Acta Chimica Slovenica, 2016
52016
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