| Identifying the proteins to which small-molecule probes and drugs bind in cells SE Ong, M Schenone, AA Margolin, X Li, K Do, MK Doud, DR Mani, ... Proceedings of the National Academy of Sciences 106 (12), 4617-4622, 2009 | 375 | 2009 |
| An aldol-based build/couple/pair strategy for the synthesis of medium-and large-sized rings: discovery of macrocyclic histone deacetylase inhibitors LA Marcaurelle, E Comer, S Dandapani, JR Duvall, B Gerard, S Kesavan, ... Journal of the American Chemical Society 132 (47), 16962-16976, 2010 | 226 | 2010 |
| Grand challenge commentary: Accessing new chemical space for'undruggable'targets S Dandapani, LA Marcaurelle Nature chemical biology 6 (12), 861-863, 2010 | 219 | 2010 |
| Homogeneous glycopeptides and glycoproteins for biological investigation MJ Grogan, MR Pratt, LA Marcaurelle, CR Bertozzi Annual review of biochemistry 71 (1), 593-634, 2002 | 211 | 2002 |
| Current strategies for diversity-oriented synthesis S Dandapani, LA Marcaurelle Current opinion in chemical biology 14 (3), 362-370, 2010 | 181 | 2010 |
| New directions in the synthesis of glycopeptide mimetics LA Marcaurelle, CR Bertozzi Chemistry–A European Journal 5 (5), 1384-1390, 1999 | 172 | 1999 |
| Aminooxy-, hydrazide-, and thiosemicarbazide-functionalized saccharides: versatile reagents for glycoconjugate synthesis EC Rodriguez, LA Marcaurelle, CR Bertozzi The Journal of organic chemistry 63 (21), 7134-7135, 1998 | 151 | 1998 |
| Chemical synthesis of lymphotactin: a glycosylated chemokine with a C‐terminal mucin‐like domain LA Marcaurelle, LS Mizoue, J Wilken, L Oldham, SBH Kent, TM Handel, ... Chemistry–A European Journal 7 (5), 1129-1132, 2001 | 130 | 2001 |
| Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries JT Lowe, MD Lee IV, LB Akella, E Davoine, EJ Donckele, L Durak, ... The Journal of organic chemistry 77 (17), 7187-7211, 2012 | 120 | 2012 |
| Synthesis of Oxime-Linked Mucin Mimics Containing the Tumor-Related TN and Sialyl TN Antigens LA Marcaurelle, Y Shin, S Goon, CR Bertozzi Organic Letters 3 (23), 3691-3694, 2001 | 108 | 2001 |
| Linear synthesis of the tumor-associated carbohydrate antigens Globo-H, SSEA-3, and Gb3 F Bosse, LA Marcaurelle, PH Seeberger The Journal of Organic Chemistry 67 (19), 6659-6670, 2002 | 93 | 2002 |
| DNA-encoded chemical libraries AL Satz, A Brunschweiger, ME Flanagan, A Gloger, NJV Hansen, L Kuai, ... Nature Reviews Methods Primers 2 (1), 3, 2022 | 90 | 2022 |
| Chemoselective Elaboration of O-Linked Glycopeptide Mimetics by Alkylation of 3-ThioGalNAc LA Marcaurelle, CR Bertozzi Journal of the American Chemical Society 123 (8), 1587-1595, 2001 | 88 | 2001 |
| Synthesis of an oxime-linked neoglycopeptide with glycosylation-dependent activity similar to its native counterpart LA Marcaurelle, EC Rodriguez, CR Bertozzi Tetrahedron letters 39 (46), 8417-8420, 1998 | 83 | 1998 |
| Recent advances in the chemical synthesis of mucin-like glycoproteins LA Marcaurelle, CR Bertozzi Glycobiology 12 (6), 69R-77R, 2002 | 78 | 2002 |
| Diversity-oriented synthesis yields a novel lead for the treatment of malaria RW Heidebrecht Jr, C Mulrooney, CP Austin, RH Barker Jr, JA Beaudoin, ... ACS medicinal chemistry letters 3 (2), 112-117, 2012 | 72 | 2012 |
| Application of natural product-inspired diversity-oriented synthesis to drug discovery LA Marcaurelle, CW Johannes Natural Compounds as Drugs: Volume II, 187-216, 2008 | 72 | 2008 |
| Combinatorial carbohydrate chemistry LA Marcaurelle, PH Seeberger Current opinion in chemical biology 6 (3), 289-296, 2002 | 71 | 2002 |
| Accessing Skeletal Diversity Using Catalyst Control: Formation of n and n + 1 Macrocyclic Triazole Rings AR Kelly, J Wei, S Kesavan, JC Marie, N Windmon, DW Young, ... Organic letters 11 (11), 2257-2260, 2009 | 69 | 2009 |
| Diversity-oriented synthesis of a cytisine-inspired pyridone library leading to the discovery of novel inhibitors of Bcl-2 LA Marcaurelle, C Johannes, D Yohannes, BP Tillotson, D Mann Bioorganic & medicinal chemistry letters 19 (9), 2500-2503, 2009 | 57 | 2009 |
