Synthesis and anticonvulsant activity of 6-methyl-2-thioxo-2, 3-dihydropyrimidin-4 (1H)-one acetamides H Severina, O Skupa, A Khairulin, N Voloshchuk, V Georgiyants Journal of Applied Pharmaceutical Science 9 (2), 12-19, 2019 | 19 | 2019 |
Synthesis, in vivo and in silico anticonvulsant activity studies of new derivatives of 2-(2, 4-dioxo-1, 4-dihydroquinazolin-3 (2H)-yl) acetamide WM El Kayal, SY Shtrygol, SV Zalevskyi, A abu Shark, VV Tsyvunin, ... European journal of medicinal chemistry 180, 134-142, 2019 | 16 | 2019 |
Synthesis, docking study, and pharmacological evaluation of S-acetamide derivatives of 4, 6-dimethyl-2-thiopyrimidine as anticonvulsant agents HI Severina, OO Skupa, NI Voloshchuk, VA Georgiyants Journal of Applied Pharmaceutical Science 10 (07), 001-008, 2020 | 13 | 2020 |
Synthesis and anticonvulsant activity of 6-methyl-2-((2-oxo-2-arylethyl) thio) pyrimidin-4 (3 H)-one derivatives and products of their cyclization HI Severina, OO Skupa, NI Voloshchuk, MM Suleiman, VA Georgiyants Pharmacia 66, 141, 2019 | 11 | 2019 |
Design, Synthesis and In Vitro Antimicrobial Activity of 6-(1H-Benzimidazol-2-yl)-3, 5-dimethyl-4-oxo-2-thio-3, 4-dihydrothieno [2, 3-d] pyrimidines SV Vlasov, OD Vlasova, HI Severina, KY Krolenko, OV Borysov, ... Scientia Pharmaceutica 89 (4), 49, 2021 | 10 | 2021 |
The Synthesis and In Silico Antihypertensive Activity Prognosis of New Mannich Bases Containing the 1, 2, 4-Triazole Moiety L Perekhoda, V Georgiyants, H Yeromina, I Drapak, V Lubenets, ... Chemistry 14 (2), 214-220, 0 | 10 | |
Synthesis and alkylation of 1-aryl-1, 5-dihydro-4H-pyrazolo [3, 4-d] pyrimidin-4-ones as possible anticonvulsant agents AI Severina, VA Georgiyants, SY Shtrygol, DA Kavraiskyi Scholars Research Library, 2015 | 8 | 2015 |
Synthesis and anticonvulsant activity of new 2-(4-oxo-2-thioxo-1, 4-dihydro-3 (2h)-quinazolinyl) acetamides ND Bunyatyan, HI Severina, EKW Mokhamad, SV Zalevskyi, SY Shtrygol, ... Pharmaceutical Chemistry Journal 54 (1), 1-6, 2020 | 5 | 2020 |
Synthesis of N-substituted derivatives of 1-(4-methoxyphenyl)-1, 5-dihydro-4H-pyrazolo [3, 4-d] pyrimidin-4-one as potential anticonvulsants AI Severina, VА Georgiyants, SY Shtrygol, DP Kavraiskyi | 5 | 2016 |
Molecular docking studies of N-substituted 4-methoxy-6-oxo-1-aryl-pyridazine-3-carboxamide derivatives as potential modulators of glutamate receptors HI Severina, VA Georgiyants, SM Kovalenko, NV Avdeeva, AI Yarcev, ... Research Results in Pharmacology 6, 69, 2020 | 3 | 2020 |
Experimental study of new pyrazolo [3, 4-D] pyrimidine-4-one derivatives for anticonvulsant activity spectrum ДП Каврайський, СЮ Штриголь, ВА Георгіянц, ГІ Северіна ScienceRise: Pharmaceutical Science, 10-17, 2016 | 3 | 2016 |
Скрининг противосудорожной активности новых производных пиримидин-4 (3н)-она АИ Северина, ОО Скупая, ВА Георгиянц, НИ Волощук Journal of Siberian Medical Sciences, 2013 | 3 | 2013 |
Синтез і прогноз біологічної активності нових N-арил-4-(2, 6-R-піримідин-4-тіо) ацетамідів ГІ Северіна, ОО Скупа, ВА Георгіянц Журнал органічної та фармацевтичної хімії, 2012 | 3 | 2012 |
Синтез, фізико-хімічні властивості та прогноз фармакологічної активності нових похідних 2-ізопропіл-5, 6-R-піримідин-4 (3Н)-ону ГІ Северіна, ОО Скупа, ВА Георгіянц Фармацевтичний журнал, 54-59, 2011 | 3 | 2011 |
Design, Synthesis, In Vivo and In Silico Anticonvulsant Activity Studies of Derivatives of 6-Amino-4-Hydroxy-2-Thio-Pyrimidine HI Severina, OO Skupa, NI Voloshchuk, AR Khairulin, VA Georgiyants ACTA Pharmaceutica Sciencia 58 (3), 0 | 3* | |
Synthesis and Antimicrobial Evaluation of 2-(6-Imidazo [1, 2-a] pyridin-2-yl-5-methyl-2, 4-dioxo-3-phenyl-3, 4-dihydrothieno [2, 3-d] pyrimidin-1 (2H)-yl)-N-arylacetamide … SV Vlasov, HI Severina, OV Borysov, KY Krolenko, PE Shynkarenko, ... Molbank 2022 (1), M1331, 2022 | 2 | 2022 |
Development and validation of hplc determination of related substances in a novel anticonvulsant agent epimidin HI Severina, SM Gubar, IV Bezruk, AS Materiienko, L Ivanauskas, ... Research Journal of Pharmacy and Technology 14 (6), 3223-3231, 2021 | 2 | 2021 |
Design, synthesis, molecular docking and anticonvulsant evaluation of 6-methyl-2-arylaminopyrimidin-4 (3H)-one H Severina, N Voloshchuk, N Saidov, V Georgiyants Severina, H., Voloshchuk, N., Saidov, N., Georgiyants 2020, 9-17, 2020 | 2 | 2020 |
Dependence of anticonvulsant activity of 1-aryl-1, 5-dihydro-4H-pyrazole [3, 4-d] pyrimidine-4-one derivatives on biopharmaceutical factors AI Severina, DP Kavraiskyi, IV Kovalevska, SY Shtrygol, EA Ruban, ... | 2 | 2017 |
Development of HPLC method for quantitative determination of epimidin-new perspective АPhI with anticonvulsive activity H Severina, I Bezruk, L Ivanauskas, V Georgiyants ScienceRise: Pharmaceutical Science, 4-11, 2020 | 1 | 2020 |