Підписатись
Yevheniia Velihina
Yevheniia Velihina
PhD Student, Engineer, V.P. Kukhar Institute of Bioorganic Chemistry and Petrochemistry of the
Підтверджена електронна адреса в bpci.kiev.ua - Домашня сторінка
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Посилання
Рік
Synthesis, in silico and in vitro Evaluation of Novel Oxazolopyrimidines as Promising Anticancer Agents
Y Velihina, T Scattolin, D Bondar, S Pil'o, N Obernikhina, O Kachkovskyi, ...
Helvetica Chimica Acta 103 (12), e2000169, 2020
142020
Intrinsic drug potential of oxazolo[5,4‐d]pyrimidines and oxazolo[4,5‐d]pyrimidines
VV Zhirnov, YS Velihina, OP Mitiukhin, VS Brovarets
Chemical Biology & Drug Design 98 (4), 561-581, 2021
102021
2-(Dichloromethyl) pyrazolo [1, 5-a][1, 3, 5] triazines: synthesis and anticancer activity
YS Velihina, SG Pil’o, VS Zyabrev, VS Moskvina, OV Shablykina, ...
Biopolymers & Cell 36 (1), 60, 2020
82020
Synthesis, characterization, and in vitro anticancer evaluation of 7-(1, 4-diazepan)-substituted [1, 3] oxazolo [4, 5-d] pyrimidines
YS Velihina, MV Kachaeva, SG Pilyo, OP Mitiukhin, VV Zhirnov, ...
Chem. Res. J 3, 81-93, 2018
72018
Synthesis, Characterization, and In vitro Anticancer Evaluation of 7-Piperazin-Substituted [1,3]Oxazolo[4,5-D]Pyrimidines
VSB Yevgeniya S Velihina, Maryna V Kachaeva, Stepan G Pilyo, Victor V Zhirnov
Der Pharma Chemica 10 (9), 1-10, 2018
62018
Evaluation of Anticancer Activity of 1,3‐Oxazol‐4‐ylphosphonium Salts in Vitro
M Brusnakov, O Golovchenko, Y Velihina, O Liavynets, V Zhirnov, ...
ChemMedChem 17 (20), e202200319, 2022
52022
Synthesis, electronic structure and anti-cancer activity of the phenyl substituted pyrazolo [1, 5-a][1, 3, 5] triazines
ES Velihina, NV Obernikhina, SG Pilyo, OD Kachkovsky, VS Brovarets
Current Organic Chemistry 25 (12), 1441-1454, 2021
52021
Synthesis and Evaluation of the Antiviral Activity of 2-(Dichloromethyl)pyrazolo[1,5-a][1,3,5]triazines
VSB Ye.S. Velihina, S.G. Pil’o, V.S. Zyabrev
Reports of the National Academy of Sciences of Ukraine 7, 75-80, 2019
4*2019
1,3-Oxazol-4-ylphosphonium salts as new non-peptide inhibitors of furin
VSB T.V. Osadchuk, V.K. Kibirev, O.V. Shybyryn, A.V. Semyroz, Ye.S. Velihina ...
Ukr. Biochem. J. 91 (4), 5-16, 2019
42019
SYNTHESIS OF 4-HETARYL-2-(DICHLOROMETHYL) PYRAZOLO [1, 5-a][1, 3, 5]-TRIAZINES
Y Velihina, M Kachaeva, S Pil'o, V Moskvina, O Shablykina, V Brovarets
Ukrainian Chemistry Journal 86 (5), 53-62, 2020
22020
Synthesis, Characterization and in vitro Anticancer Evaluation of 5‐Sulfinyl (sulfonyl)‐4‐arylsulfonyl‐Substituted 1, 3‐Oxazoles
V Zyabrev, S Pilyo, B Demydchuk, M Kachaeva, I Semenyuta, V Zhirnov, ...
ChemMedChem 18 (14), e202300161, 2023
12023
In silico study the interaction of heterocyclic bases with peptide moieties of proteins in “fragment-to-fragment” approach
Y Velihina, N Obernikhina, S Pilyo, M Kachaeva, O Kachkovsky
Ukrainica Bioorganica Acta, 2021
12021
In silico study of binding affinity of nitrogenous bicyclic heterocycles: fragment-to-fragment approach
YS Velihina, NV Obernikhina, SG Pilyo, MV Kachaeva, OD Kachkovsky, ...
Ukrainica bioorganica acta 15 (2), 49-59, 2020
12020
SYNTHESIS OF PYRAZOLO [1, 5-a][1, 3, 5] TRIAZINE AND OXAZOLO [4, 5-d] PYRIMIDINE DERIVATIVES AND STUDY OF THEIR VASODILATOR ACTIVITY.
YS Velihina, SG Pilyo, IV Ivanova, VS Brovarets
Issues of Chemistry & Chemical Technology/Voprosy Khimii & Khimicheskoi …, 2023
2023
Design, synthesis and evaluation of the anti-breast cancer activity of 1, 3-oxazolo [4, 5-d] pyrimidine and 1, 3-oxazolo [5, 4-d] pyrimidine derivatives
Y Velihina, R Gesese, V Zhirnov, O Kobzar, B Bui, S Pilyo, A Vovk, ...
RSC Medicinal Chemistry 14 (4), 692-699, 2023
2023
Synthesis of some oxazolo [4, 5-d] pyrimidine derivatives and evaluation of their antiviral activity and cytotoxicity
Y Velihina, S Pilʹo, O Kobzar, O Zaliavska, MN Prichard, SH James, ...
ARKIVOC: Online Journal of Organic Chemistry 2022, 2022
2022
Investigation in the fragment-to-fragment approach of the interaction of heterocyclic bases with peptide bonds of proteins
Y Velihina, N Obernikhina, O Kachkovsky, V Brovarets
Біоактивні сполуки, нові речовини і матеріали, 2021
2021
In vitro and іn silico estimation of pyrazolo [1, 5-a][1, 3, 5] triazines
Y Velihina, N Obernikhina, I Semenyuta, S Pilyo, O Kachkovsky, ...
Записки Української науково-дослідницької асоціації: тези доповідей …, 2021
2021
Взаємодія 2-ациламіно-3, 3-дихлороакрилонітрилів з 5-амінопіразолами.
YS Velihina, ER Abdurakhmanova, MV Kachaieva, SH Pilo
Хімічні проблеми сьогодення, 135-135, 2018
2018
Квантово-хімічна оцінка донорно-акцепторних властивостей азотовмісних спряжених гетероциклів
ЄС Велігіна, МВ Качаєва, НВ Оберніхіна, СГ Пільо, ОД Качковський, ...
Матеріали V Міжнародної науково-практичної конференції молодих учених …, 2018
2018
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